No. |
Title |
Author(s) |
Downloads
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01 |
A Tribute to Prof. Vincenzo Tortorella
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Girolamo Cirrincione |
PDF
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02 |
H-NMR determination of the enantiomeric excess of the antiarrhytmic drug Mexiletine by using mandelic acid analogues as chiral solvating agents
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Giuseppe Carbonara; Alessia Carocci; Giuseppe Fracchiolla; Carlo Franchini; Giovanni Lentini; Fulvio Loiodice; Paolo Tortorella |
PDF
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03 |
Synthetic approaches to difluoroindolecarboxylic acid ethyl esters
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Romano Silvestri; Marino Artico; Giuseppe La Regina; Gabriella De Martino |
PDF
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04 |
Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents
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Antonello Mai; Marino Artico; Sergio Valente; Ilaria Cerbara; Olivia Befani; Paola Turini Laura Dalla Vedova; Enzo Agostinelli |
PDF
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05 |
Synthesis and pharmacological evaluation of 7-substituted 1-ethyl-3,4,10-trimethyl-1,10-dihydro-11H-pyrazolo[3,4-c][1,6]benzodiazocin-11-one. A new ring system
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Onofrio Migliara; Salvatore Plescia; Patrizia Diana; Vita Di Stefano; Lorenzo Camarda; Roberta Dall’Olio |
PDF
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06 |
Glyceroglycolipids from Euphorbia nicaeensis All. with antiinflamatory activity
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Francesca Cateni; Gioacchino Falsone; Jelena Zilic; Paolo Bonivento; Marina Zacchigna; Dušan Žigon; Silvio Sosa; Gianmario Altinier |
PDF
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07 |
A new synthesis of triazolo[4,5-g]quinolines and unexpected ring reduced products by treatment with hydrazine hydrate
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Antonio Carta; Giuseppe Paglietti |
PDF
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08 |
2-[(E)-3-(6-chloroimidazo[2,1-b]thiazol-5-yl)prop-2-enyl]-5,6-dimethoxy-3-methyl-1,4-benzoquinone: a new inhibitor of NADH dehydrogenase with antitumor activity
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Aldo Andreani; Massimiliano Granaiola; Alberto Leoni; Alessandra Locatelli; Rita Morigi; Mirella Rambaldi; Giorgio Lenaz; Romana Fato; Christian Bergamini |
PDF
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09 |
Synthesis of new pyrido[4,3- g and 3,4- g]quinoline-9,10-dione and dihydrothieno[2,3- g and 3,2-g]quinoline-4,9-dione derivatives and preliminary evaluation of cytotoxic activity
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Isabel Gomez-Monterrey; Pietro Campiglia; Teresa Lama; Paolo La Colla; Maria V. Diurno; Paolo Grieco; Ettore Novellino |
PDF
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10 |
Synthesis of pyrrol-[1,2-a]indole-1,8(5H)-diones as new synthones for developing novel tryciclic compounds of pharmaceutical interest
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Mario Sechi; Alessio Mura; Luciano Sannia; Maria Orecchioni; Giuseppe Paglietti |
PDF
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11 |
Molecular modeling of β-cyclodextrin inclusion complexes with pharmaceutical compounds
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Stefano Alcaro; Danilo Battaglia; Francesco Ortuso |
PDF
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12 |
Synthesis and biological evaluation of 3-alkyloxazolidin-2-ones as reversible MAO inhibitors
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Claudia Lamanna; Maria Stefania Sinicropi; Paola Pietrangeli; Filomena Corbo; Carlo Franchini; Bruno Mondovì; Antonio Scilimati |
PDF
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13 |
Methyl derivatives of tetracyclic psoralen analogues: antiproliferative activity and interaction with DNA
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Lisa Dalla Via; Eugenio Uriarte; Lourdes Santana; Sebastiano Marciani Magno; Ornella Gia |
PDF
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14 |
Microwave-induced synthesis of benzimidazole and thiazolidinone derivatives as HIV-1 RT inhibitors
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Angela Rao; Alba Chimirri; Stefania Ferro; Anna Maria Monforte; Pietro Monforte; Maria Zappalà |
PDF
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15 |
1-Phenyl-3-azabicyclo[3.1.0]hexane derivatives as new ligands for sigma receptors
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Agostino Marrazzo; Andrea Pappalardo; Orazio Prezzavento; Franco Vittorio |
PDF
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16 |
Synthesis and anticonvulsant properties of 1,2,3,4-tetrahydroisoquinolin-1-ones
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Rosaria Gitto; Maria L. Barreca; Eleonora Francica; Roberta Caruso; Laura De Luca; Emilio Russo; Giovambattista De Sarro; Alba Chimirri |
PDF
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17 |
A general, versatile synthesis of 2H-pyrrolo[3,4-c]quinolines via tosylmethylisocyanide reaction
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Roberto Di Santo; Roberta Costi; Michela Forte; Carlo Galeffi |
PDF
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18 |
Synthesis of 5-substituted 7,9-dihydro-8H-[1,3]dioxolo[4,5-h][2,3]benzodiazepin-8-ones as anticonvulsant agents
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Maria Zappalà; Nicola Micale; Silvana Grasso; Frank S. Menniti; Giovambattista De Sarro; Carlo De Micheli |
PDF
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19 |
Aminoacyl-analogues of mitoxantrone as novel DNA-damaging cytotoxic agents
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Giuseppe Zagotto; Claudia Sissi; Barbara Gatto; Manlio Palumbo |
PDF
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20 |
DNA-binding and DNA-photocleavaging properties of 12a,14a-diazoniapentaphene
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Giampietro Viola; Heiko Ihmels; Hubert Kraußer; Daniela Vedaldi; Francesco Dall’Acqua |
PDF
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21 |
Antifungal and antimycobacterial activity of new N1-[1-aryl-2-(1H-Imidazol-1-yl and 1H-1,2,4-triazol-1-yl)-ethylidene]-pyridine-2-carboxamidrazone derivatives: A combined experimental and computational approach.
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Maria Grazia Mamolo; Daniele Zampieri; Valeria Falagiani; Luciano Vio; Maurizio Fermeglia; Marco Ferrone; Sabrina Pricl; Elena Banfi; and Giuditta Scialinoc |
PDF
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22 |
H-NMR and FT-IR study of the state of melatonin confined in membrane models: location and interactions of melatonin in water free lecithin and AOT reversed micelles
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David Bongiorno; Leopoldo Ceraulo; Mirella Ferrugia; Felice Filizzola; Cristina Giordano; Angela Ruggirello; Vincenzo Turco Liveri |
PDF
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23 |
Docking of indolo- and pyrrolo-pyrimidines to DNA. New DNA-interactive polycycles from amino-indoles/pyrroles and BMMA
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Antonino Lauria; Patrizia Diana; Paola Barraja; Alessandra Montalbano; Gaetano Dattolo; Girolamo Cirrincione; Anna Maria Almerico |
PDF
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24 |
Synthesis of potential dual binding site acetylcholinesterase inhibitors through an efficient solid phase approach based on the Mitsunobu reaction
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Francesco Leonetti; Anna Cappa; Cristina Maccallini; Angelo Carotti |
PDF
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25 |
Design, synthesis and preliminary pharmacological evaluation of rigid analogues of the nicotinic agonist 1,1-dimethyl-4-phenylpiperazinium iodide (DMPP)
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Luca Guandalini; Elisabetta Martini; Fulvio Gualtieri; M. Novella Romanelli; Katia Varani |
PDF
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26 |
Adenosine receptor agonists: synthesis and binding affinity of 2- (aryl)alkylthioadenosine derivatives
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R. Volpini; S. Costanzi; C. Lambertucci; F. R. Portino; S. Taffi; S. Vittori; K.-N. Klotz; G. Cristalli |
PDF
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27 |
Synthesis of new 5-phenyl[1,2,4]triazole derivatives as ligands for the 5-HT1A serotonin receptor
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Loredana Salerno; Mariangela Siracusa; Francesco Guerrera; Giuseppe Romeo; Valeria Pittalà; Maria Modica; Tiziana Mennini; Filippo Russo |
PDF
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28 |
β-Aminomethylation of N-aryl- and N-azaheteroaryl-substituted methyl 2,5-dimethylpyrrole-3-carboxylates. Kinetic effect of the N-pyrrole substituent
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Mariangela Biava; Giulio Cesare Porretta; Giorgio Giorgi; Giancarlo Sleiter |
PDF
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29 |
9-Fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II
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Stefano Alcaro; Adriana Arena; Rosaria Di Bella; Simonetta Neri; Rosaria Ottanà; Francesco Ortuso; Bernadette Pavone; Maria Gabriella Vigorita |
PDF
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30 |
Solid phase synthesis of 5,6-disubstituted pyrimidinone and pyrimidindione derivatives
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Maria Cristina Parlato; Claudia Mugnaini; Michela Lucia Renzulli; Federico Corelli; Maurizio Botta |
PDF
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31 |
Aromatic Schiff bases and 2,3-disubstituted-1,3-thiazolidin-4-one derivatives as antiinflammatory agents
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Iana Vazzana; Emanuela Terranova; Francesca Mattioli; Fabio Sparatore |
PDF
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32 |
Dynamic kinetic resolution of alpha-bromoesters containing lactamides as chiral auxiliaries
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Alessandra Ammazzalorso; Rosa Amoroso; Giancarlo Bettoni; Barbara De Filippis; Letizia Giampietro; Cristina Maccallini; Maria Luisa Tricca |
PDF
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33 |
A step further in the discovery of phthalein derivatives as Thymidylate Synthase inhibitors
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Samuele Calò; Donatella Tondi; Alberto Venturelli; Stefania Ferrari; Piergiorgio Pecorari; Marcella Rinaldi; Stefano Ghelli; M. Paola Costi |
PDF
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